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Luhman J.1990, A New species of Aphidius (Hym.) attacking the pea aphid, 
Acyrthosiphon pisum. Emtomonphagus, 35(4):509-514]λѧ
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УסޣŽҲʵܣָͽŽ
ΪŽڵĲʿл Tiagabine ĺϳоͬʱŽ߻
һʿҲڸʵGABA תƼоϺпίĿ
ȷǸѧҩѧԺоһʿĳɹɼ
BMCL йҩﻯѧ־£ԺʿûоָBMCL 
Ϊ˫ҲԺʿлJianbin Zheng, Ren Wen*, 
Xiaomin Luo, Guoqiang Lin, Jiange Zhang, Linfeng Xu, Lihe Guo, 
Huangliang Jiang. Design, synthesis and biological evaluation of the 
N-diarylalkenyl-piperidine carboxylic acid derivatives as GABA uptake 
inhibitors (I). Bioorganic & Medicinal Chemistry Letters. 2006  16(1): 
225-227Ժʿʵ˿⿪ʼʱԺʿһʿŽ
ӣֻŽһˡŽʵԶĿϺпί
ؿӿĿĿȷд֪ʶȨɺ
й˫ǰֹǿԺʿǳҲӦóʵ

2) Ž"ʱ걨ϺпίصĿʱϺл
ʿģûоԴտ˲ùأӦ͵ֹ
ǿоԱæ뵽Ŀ20 "

ͽڴĿҪʵʩڼ䲢Žû20 
˹˹ءʵŽлʱͬʱĿڸ
ҩѧԺչһֱǰнÿλʦѧеȸ
ƶȣû20 򾭷ѣʵʵλ18 򣩣
Ŀѧд̲ġרоָȵȹ
ӦɵĹŽڸŽԺŽ˻
18 ӦѧУˣȫʵġ⵱ʱŽ֮
ȥлҲչϣӿɵһ֪ĺϳɺ
о⣨ԭ˶ʿĿ⣩תGABA תƼоĺ
ⶼ֪ṹ֪·߷Ŀ껯Ϊ
ȱѧҪףҩ˶֪ͨȡ̣
ԡײĵȷŽĻŰʵߵ
ˣŽڵĺⶼĨˣԺʿŽֺ

3) Ž˵"оûκιסֻϵĵʦ
оϺлʵʩġ"

˿л͸Ϻί⣬ŽǴѧ
ͽڿ鵽лʵģʵ¼дڸѧҷĸ
ѧʵ¼ϣɵѧУҺʵйطҩGABA ת
ƼTiagabine ĺϳɷо棬õԺʿİָ
ҲδлĹ׺ԺʿָͬһŽ﷢ڡй
ѧ챨Jiange Zhang, Changsheng Jiang, Guoqiang Lin*, Ren Wen*. A 
New Synthesis of 4, 4-Diaryl/Diheteroaryl-3-butenyl Derivatives of 
Nipecotic Acids as GABA Transporter Inhibitors. Chinese Chemical 
Letters. 2005  16(9), 1205-1208 ͡ߵѧУѧоJian-ge 
Zhang, Changsheng Jiang, Jianbin Zheng, Ren Wen*, Guoqiang Lin*. A new 
synthesis method and GABA transporters inhibitory activities of 
tiagabine and its analogues. Chemical Research in Chinese Universities. 
2006  22(3): 351-355 оֹǿ˫ͨѶߣ
GABA תƼTiagabineṹ½ṹơϳɼ
Է˼·⼰о·ߵȷ棬ҪŽڸġ
Žÿ1-2ܶҪμŽڿСᣬŽڵѧһ
ڻϻ㱨ڹչȻȡŽڵָŽڼ
ԱʱŽ»ƺͺϳҲཨԵ
ͽ顣»ʱŽڸٵĲοףоͰ
˺ BMCL˼йصϡ BMCL漰ĺ򻯺˼
ҲŽڸ׽ӵԭҩﻯѧĻۣ
ġҵʱŽﻹʱʱڿϱԹԺʿ»Ȥֻ
Ž Tiagabine ƱϳɡŽڿǵŽﲩʿҵľ
ҪΪ»ԺʿԵһλЭ̣
ҩﻯѧлѧҪͬΪոѧҩﻯѧʿо
ҪȥҪ൱»ԼֲʿĵĴԣ
ŽڵʱлоĿγ̽ѧÿܶҪȥлϿΣκ
ŽڻȥлŽڵʵҿʵΪ˰
ɿ⣬ʱҵȺѧƱҵкϳɣÿ
һѧڱҵĹлѧרȥлϳԭϵġ
Ž֣ݴѧ˶ʿоܹʸǶŽоָͰ
ĵʦŽʸǸЦ BMCL оŽ
2005 격ʿҵǰȫɣе˶ʿκιϵ
ϸ̸

֪˶֪Ž˶ʿʱĻ˶Ž
ͳŵ˱ʾȫ֧Žڲͬģ˺Žһֱȫ
˳ͨ˶ԺоȣֱĴ硣
ڿŽ˵мСأѧпնŽ
ĵĿγѧϰʵѵͺڵѡ⿪ڿ˺оȶõ
ŽڵϤָͰŽﲩʿĵĿҲŽڷ
ȷģƪĶŽڵĶξ޸ģν渺Ž
ղʿĴҲŽֵġŽоϣѧ
ǼǱγѧϰɼоǼǱⱨ棬ڿˣҵǼǱ
оֲᣬĴĴίԱἰ飬ѧλ
ԭʼ¼㱨¼ȣȷдŽĵʦŽ
ǩָʵҲĿáΪŽָСԱԺʿȴ
ơ⡢ڿˡ޸ԼĿȷȴδκ
飬ҲδμŽĲʿĴ硣ŽΪ"ϵ"
ʦѾǳְˣоϺлģŽ
ںαô档

4) Ž˵"ұҵǰⷽоտʼдо
ֽڵȨ½˲ֹתңҼ¸÷о
оظһЩؼʵ飬ڴ˻ϣл򻯺ĺϳ
оЩоĻϣ2006 ˹Ȼѧ
һ˹ȻѧС"

Žԣĵ BMCLӦ
ʿҵĳɹܿϧ䲩ʿѧλ BMCL ĺδ
κһ»2005ҵĳɹֻȫհ䲩ʿ
Ľν"ҵоظһЩؼʵ"ʵǿؼû
κµĶҲȥŽ"ԺʿȨ˲ֹת"
Ƿȷ˿Ǹѧлͬĺ⣩
֣ݴѧ˶ʿоΪ˵١
Ȼһ֪Ž 2005ҵȥʿһ꣬ڸ
ҩѧԺ¼½ҩҪȥҮ³ѧߣʱ;л
򻯺ĺϳоȻֻܽǰΪѧʿоʱ
ð 2007 꿪ʼʵʩĹȻѧоɹԽʳ

5) Ž˵"ڽоĹУ֣ݴѧУʡƼ
лԺʿϣ֧ҵĹ"

ŽĻȫ¶ҹĿǰȻѧȹҼĴ
⣬ЩֻҪ㶨˸λϵĹؼ""һ·˳˳ˮ˳
¿⣬νóϧŽ̫ڼ
Ŀƽ𡢴о󡣽ֻܰԭѧʿоڼ
о¶ţҲö""֣ݴѧУ
ʡƼԺʿǺòΣŽһִ绰Žͨ
ǲܵģҲֻǿʶƱ絽סĹؼֻаѸѧ
ڳ׷񶨣ܰԭڸѧǲ֪ʶȨ͵͵鵽֣ݴѧ
ǸȻѧ£ŴͨЩѾһ
Ŀ

6) Ž˵"˶ӵ£ʹָµ˶ʿоδȡ
ʵԽչлȡýչʱŽװǡ"

ŽڵѧˮƽΣ˽ҩﻯѧ˶ǳˣŽ
ԴŽҲվסŵġǶоǲоָӦ
öᣬ 5 ҩ˶-ѧϰǰ
ʱڿչ̫˳ҲоѧϰĿ͹۹ɵĽǰ
ѧϰѧλγ̼ϣѧϰʵ鼼ܡǿײķͿ
ڵ͹ؼӦͻƽ׶ΣҪԺһſһ
ĽʱŻнϴĲŽһ͹۹ɣǰ׶ο
չŽʵҵˮƽ͡Լԭ˼ά
ôŽڵѧȥлǷͱϲҵ
أ

7) Ž˵"ҲʿͷҪҰܷĶ
д£ҲЩǷ죬Ҫڴһϵ7 
ǰ"

νǿڴһϵ 7ǰɵʵǲġʵ
Žڵʱ֪ŽڱҵǰԺʿͺʡ쵼νк
ݣһֱŽܹģûκν䱸ģŽԼ
֡ʵǣŽڿǵѧУһ·Ժõѧλ֤
Ҫ󣬶ҩķʱҪԽȣҪ
оҵǰڷ˴ﵽԤҪ󣬾ȡڴ磬
ѧͿ԰õѧλ֤顣Žڳ˵Լʱ²ף
ϣѧʵʱģֻҪǦӡľУѧԼǱҪ
ܽᣬԺûодˡЩоҵˣڵҵǰ
Ҳ׼ĳ壬ûŽҲûԼ
ǿ޸ķʦһֱѧһߣѧ
췢չϵλⲩʿȡʱŽҵ
мλдʦƼʿҵȥʿʦ뵽
Ž뷽跨ϵҵŽʦûϵ
˵ȥƴѧʱͱʾԸȥƼһʿҵȥ
ˡ鶼֪Žڶѧҵϸģַǳѧġ
ŽΪŽڱ"лĿгɹ"ʱ֪Ž
Ұģôҩѧѧ༭޸ȫԲ
ŽԼ޻أ·Ǿ⣬Ҳн۵¼
ŽŽδ޸Ķƪҩѧѧ£˵ıⲢ
""ƪ¡

8) Ž˵"Ըѧй涨ʦΪڣӲҪҰ
ǿоԱӻڸһָСԱڸǸ
ѧѧԺְҲ֪ҵкν
ѵǿĿѧ"

ѧ涨ֻһʦŽںԺʿۺʱŽ
лԺʿʵʵ֮ǰѾʹ˵ԺʿͨԺʿ󷽵
ʾ⣬⣬ŽڻemailԺʿŽĹɹ
չľ彨飬ԺʿҲصʾͬ⣬ЩŽڿ鶼
£Ž߹ͨҲδӳŽﲩʿĵʦͽڣ
ָСԱͽڡֹǿоԱڸоԱǴδ˵
ʦǵʦ˵90ڸоԱͲŽڿ鹤
ЭɸѡҩзָŽ2000˶ʿѧʱ
ʦδݣһҽʦΪŽָСԱǶ
ĹйָϹģʦѧˣŽת
ԺָСлоԱ֡ͬʱҲŽԸ
ʦдȥģʲôǿӽȥġڷ˵ˣ
ǣǿᡣͬʱʦںģĿ
¿мƪһƪΪ6-7ߣ
﷢УʦδҲδ˵Ž
ʦּӵBMCLе˵ҲĳЩŽںͻ
ʦĨڡ

9) Ž˵"֣ݴѧ˶ʿѧʱԭҽƴѧίд
ְо"

ŽﵽΪֹı˵ѧŽǺҽ
ѧ֣ݴѧίϺҽƴѧ븴ѧĶо
ڸѧоԺȫѧ鸴ѧоԺо
Ժ浵ĸ֤ļƻγѧϰƻȣо֤ʵݡ
оڼйصплͳɹڸѧ쵼ºŽָ
º֧Ͱŵġί෽ǸѧΪһλӵвʿѧλ
ʦӵڸѧ֪ʶȨ

϶֪ʵϣҿĽ㣬Ž
˲ҪرЩԷ磬ӭָ

(XYS20070809)

˿(www.xys.org)(xys.dxiong.com)(xys.freedns.us)(xys-reader.org)

ԡĲʿǳ-Ž-ֹǿһһͣŽ
ʦĿ⡷Ĳ

ߣ˵

ϺҽƴѧָѧҩѧԺϳҩҵְҲ
ͽڵ˶ʿŲʿ2000-2002ͬһʵҹ¹
ϿλۼѵۣбҪҲһ¸˵ļ⣬
вָλָͬʱҲϣĳЩô˵¡
ҲЩMITBBSϵϣʵڲҹͬĳЩ˵ôʷʽ

˾ţ۵ĸӦǷѧˣûб
ҪŽڷѳʾһЩ֤ݣŲʿӦķ֤ʾϧǣ
ĿǰΪֹֻһЩá֮ӵĶͽƷۣʵ
ЩȤĳЩϲ£ҲòҲ˵һЩ

Һͽڹദ7꣬˵ûìܣ˵ԭ
ģ󶼿Խ˵֮䣬ĸŮ֮һ
ִĿǰΪֹҸ˶Žڵǣ齲ԭѧ淸
ǼġʱޣҪӺõһ潲
ϸʱȷ˸еѻ𡣵һҲһЩϽڵȻ
ˣǵȱ㣬ͬʱһ˵ܻ۷Լ
˱׼ڡǣҵӡͱɡª۸
ϱߣѧУͬеĿڱҲ󲻽Ī⼸
ڿʼתˣȻ˻˵ЩµĴ̰ƽʱصҲͦã
˵ûˡ

ڴˣŲʿָŽڵļ㣬ұ˾˵һ£
ɫʡ2002о뿪ҽҽ
Դǰۡ

1	֪ŽڵĿ⾭ѲǺܸԣ̫ԸӺ⣩
Ա֤ѧѧҵŲʿᵽġҺϳõʼԭȩ
ԼǮϺϳģԼǮӡġҿԸ
һֽͣݵʱѧУĲƶȣСƷ󱨡
ϰԼǮȻþѱȥҲһʱŲ
ʿҩƷ֪ΪβΪʱľѱұܣ
Լ˵ûöǮԲ뱨ˡ

׸ӡЩѧΪϲͼݣûϸ͸ӡ
ܶԿϵõףŽھͶԴ֧Щơ
ǶȫģûĳˣҸøӡĻøӡġ

2	ĸѧѧľҲ֪ǰѧѧʱһ
ҽһǲʿڿûͨڶʿԶѧģʵ
˵ҵڻûи㶮ԭ򡣵ʱŽΪʵȵԭҰʵ
顣ѧŽڻ̸Σϣټȥѧҵ
˶ʿѧʱŲʿԼҲˣʱѧҲֵͦãҺ
Ųʿһ𻹵оԺȥ˵֧ŽȰѧľ
̸ϾѾȥˣҲҪȥӰڵһѧ
ˮѧĽʦڸУ躣ҩѧƣԺԺϺˮ
ѧյġѧʱһҽѧ뿪ҽ
ãԶһЩȨġ֪ѧŽںͶԷѧ
Уһֹͬľ

ڳʵŲʿڱ˱ѧҪ˵ĵλ
ȥ֣ű˵ǴӺζġҵĹƣŽѧ
ѧͼϵʵҲܿҪ黹ѧڼʵ¼
ˡȻֻҸ˵Ĳ²⣬û֤

3	Ųʿ˶ʿڼʵȵȷԭλ֣ݴѧ
йءʱҪ˶ʱŽھʮԥ
ڽ뿪ҽ֪Žڱ֤ŬԼרҵ
ܺǶˡǵ뿪ҽʱ򣬻ŽڱʾŲʿ
һѧѧĵġǵĿǲܰڱҵȻ
ŲʿҲпܾʹ֮мߣ˶Žڵˮƽڴ
ϲˡ

4	ŲʿһЩŽһѧѧ
Ͷһ˵ҲٶۣȤĿȥһ¡Ҫ˵ǣ
Щڸԭ;ֹģŽڵѧûбڵģǰҵ
ҵ˵

(XYS20070809)

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ŽͽĽһش

ߣ֣

ŽﲩʿĶλظѻظһ£Ųʿѵһ
ھϲ½ϺáԵƺԡλظŲʿĵһ
ظԵıʣڶλظαװ

1˵Ĳʿолʦֹǿо⡱
εлǺƳȥлڸ˰æȻ
ڵоΪʲôԺʿĿ⣿м϶˵

2ⲿֹ֪ʶȨڱ²ͽС
£֪ʶȨǵλ֮飬Ϊһоֻиɻķݣ
Щ£ֱӿ϶֪ʶȨĹҪô֪ҪôƱ硣

3λظĵʵǵһļ˵һȻ


4λظĵ˵ǲʿڼĹ˼ڵ
ʦĹĻϵĹʵǵ˵ʦĿ⣬Υ

5λظĵһͬ

6֣ݴѧίо˵֪ʶȨ֣ݴѧûйϵΪ
оûڸУɡ

7λظĵֵö˵˿߽Сߡ
֪ʶȨĿŵԣɼƷ

8ѧĹ涨Ȩ鸴ѧΪһоȨ
ظ˵һ䣬֪ʶȨǵλ֮飨˳⣩ѧо
ûйϵһɻˣȨ⡣

9עѧ˵һҲˡ

10òʿûдʹڲðѲʿԼ
bmclϷʹڲڵʦǽǡ

11ԹġûдʹڡȢϱ
Լˣ˸ĸ࣡

12ұȡֶεȨȨ绰¼ûд
֤šɲɡ

󣬡Žڵڹȥļȷ͹˼Ӱ졣
ܸǣȻרעҵоԸΪ
˲¼ľ޼ִֵŽھʹµȨ
Ļͨйѧţ˾ţˣ
һ쵼ļơС¿ˮ̡ķСΡȻ
էէءĲţźŲʿǴ򣬲֪
ַѧ֪ʶȨл֪ʶȨ

о׻һãҲҲΪһţ
ˣɱ֣ݴѧֵ

ллйҡҺ֧ҵˣлû˵Ҿ
ð˵ˣЩˡ֪Է

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ˣ

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ֹǿ֮ʵʺڣ

ߣȶ

˿ϳָʲô"д"ĺɴ˵£Щź
"ռ"ĵ񺺣Ҫ黯մվ
ҶҪʵڵȻûб˵˭"д"κ¶
۵ԣ˵"д"зɡ 

룬˫ƽ͵ԷĹ۵ʵеѾ
ȴȻϣһظЩɰͰ͵Ĺ۵㣬Գʵ
ۻû壿 

ϴΰ"Žֹ֮ǿ֮ʵںη"д
"ͼ̽һЩ뷨ҵ𰸺޸İԭй۵"һЩ
ֵ˼⣬ۣ

1. ໥ִˣʦϵû˷ԣŸ
ڵ긴עᵽлĹʱҲоݣŸڶ
λζλһȷ"Ӳ"֤ݣίЭȣ
˫λ£ܿûдκ֤ݣƶǵʱֵʦ
֮Э⡣ֵʱ޴ӲڽûзԺʿָ
СԱԺʿƺŽ︱˵ֹǿʦ˵û
飬֧ŵҲŵĵʦ˵Ž︱ϻظȫ
ͬoŵĵ绰⣬ƺԺʿ
ʦݵɣȻڶţ"ʦѵİ"̬ͣ
ûзһŵˣƶλʦͬһ㣬ܾǴҹ
עĴˣ֮֮Զӷɸۣ
ԺʿҪŵݣԺʿӦЧ֤ݣĿǰԺʿӲ
֤ƺûУûеʱԸ⹫ 

2. ¶֮пкϵǷȷ
ϺίĿɴ˿ƶŽ︱ΪſԱԺʿʵ
пкʵΪкĿ;ѷ䣬֮
⡣⣬ӲǷƶԺʿṩǷҲ漰Źͬ
ĿʵõǮԺʿԼ⾭ѣŹͬĿľѣ
Ҫһ֤⣬ϣŶʵϺί
̬أ 

ûҵ´ǰ޸ԭй۵㣬ϧһЩ
֮ƶϡȻ˵"˿⽫ֽ
⡭"棬ЩˣڹⶼЦ˵ͳϰ岻
֪λԺηλ˱Žλữѧ
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˸ø, ܸоŽＫпһӲŵ.

ڡͽĽһش̸, ĵĿ, , 
˼·ȵȾл, ˵ѧŽڶ䲩ʿûһ
㹱, Žֻһ.ΪŽĲʿѧλǸѧ,
пԺл? һŽӦ˵.

֪, ˶ѧڼ, ʦ˵Լѧܷѧλо
ķȨ.ʦ,Ҳѻѧλ.˿,Ž
ѧλ֮ǰ, ϶Žڹϵǲ.ѧλѾ,ŽڶŽ
Ѿû,ΪûȨû, Ժʿͬ,ٰѾһ
.Ҫ֪һǶô.Ժʿô,Ͳͬ.Ž
пһӲŵ.

ڸûظл̸ "20068»ùȻѧĿһڵ
С8Ԫ", ӱ¶˸ûԺʿֶͨΰõ.
֪, һίÿ9ºŸ֪,8
ͻ. Ӧ֪˸.֪ӦԺʿ.

ʿѧλһƼ˵мֵһ.Žڰ.
,Լĵʦӵ϶ǲӦõ.

2007 8 9

(XYS20070809)

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¼йоĲ֮

ߣСѧ

ڱ˿¼ӦǾйɫġҲ˭˭ǣҸо
йеоǺ
ˡȥԴӦóԲоϵ¼Ǳ˵
׾

һΪʲôŲʿҪȥһʵҵģйֿѧ
˵ţëΪԼѡ˵ʦʦʽָһ
оû취ֻܰѧͳȥҪҪѧԵʦڵλΪ
巢ģ𣿱ʵҵоɹַʽλռ


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˻ᣬһҶԷľͶԸλ־ʿĸл
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¹ܿ(SPIEGEL ONLINE)
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IntroductionҲȷʵ˵Ҫһconceptual framework
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